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OpenAlex Citation Counts

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OpenAlex is a bibliographic catalogue of scientific papers, authors and institutions accessible in open access mode, named after the Library of Alexandria. It's citation coverage is excellent and I hope you will find utility in this listing of citing articles!

If you click the article title, you'll navigate to the article, as listed in CrossRef. If you click the Open Access links, you'll navigate to the "best Open Access location". Clicking the citation count will open this listing for that article. Lastly at the bottom of the page, you'll find basic pagination options.

Requested Article:

Structure-based design of targeted covalent inhibitors
Richard Lonsdale, Richard A. Ward
Chemical Society Reviews (2018) Vol. 47, Iss. 11, pp. 3816-3830
Closed Access | Times Cited: 291

Showing 51-75 of 291 citing articles:

Systematic Study of the Glutathione Reactivity of N-Phenylacrylamides: 2. Effects of Acrylamide Substitution
Adam B. Birkholz, David J. Kopecky, Laurie P. Volak, et al.
Journal of Medicinal Chemistry (2020) Vol. 63, Iss. 20, pp. 11602-11614
Closed Access | Times Cited: 51
Pooled analysis of safety data from clinical trials evaluating acalabrutinib monotherapy in mature B-cell malignancies
Richard R. Furman, John C. Byrd, Roger G. Owen, et al.
Leukemia (2021) Vol. 35, Iss. 11, pp. 3201-3211
Closed Access | Times Cited: 49
Recent Advances in BTK Inhibitors for the Treatment of Inflammatory and Autoimmune Diseases
Datong Zhang, Gong He, Fancui Meng
Molecules (2021) Vol. 26, Iss. 16, pp. 4907-4907
Open Access | Times Cited: 49
Recent progress in covalent warheads for in vivo targeting of endogenous proteins
Naoya Shindo, Akio Ojida
Bioorganic & Medicinal Chemistry (2021) Vol. 47, pp. 116386-116386
Open Access | Times Cited: 44
Site‐Selective Pyridine C−H Alkylation with Alcohols and Thiols via Single‐Electron Transfer of Frustrated Lewis Pairs
Chang‐Yin Tan, Myojeong Kim, Inyoung Park, et al.
Angewandte Chemie International Edition (2022) Vol. 61, Iss. 51
Closed Access | Times Cited: 35
Discovery of SARS-CoV-2 main protease covalent inhibitors from a DNA-encoded library selection
Rui Ge, Zuyuan Shen, Jian Yin, et al.
SLAS DISCOVERY (2022) Vol. 27, Iss. 2, pp. 79-85
Open Access | Times Cited: 34
Peptide‐based covalent inhibitors of protein–protein interactions
Felix M. Paulussen, Tom N. Grossmann
Journal of Peptide Science (2022) Vol. 29, Iss. 1
Open Access | Times Cited: 34
The expanding repertoire of covalent warheads for drug discovery
Namrashee V. Mehta, Mariam S. Degani
Drug Discovery Today (2023) Vol. 28, Iss. 12, pp. 103799-103799
Closed Access | Times Cited: 21
Chemical technology principles for selective bioconjugation of proteins and antibodies
Preeti Chauhan, V. Ragendu, Mohan Kumar, et al.
Chemical Society Reviews (2023) Vol. 53, Iss. 1, pp. 380-449
Closed Access | Times Cited: 19
Characterization of a Potent and Orally Bioavailable Lys-Covalent Inhibitor of Apoptosis Protein (IAP) Antagonist
Parima Udompholkul, Ana Garza-Granados, Giulia Alboreggia, et al.
Journal of Medicinal Chemistry (2023) Vol. 66, Iss. 12, pp. 8159-8169
Open Access | Times Cited: 18
Peptide-Based Covalent Inhibitors Bearing Mild Electrophiles to Target a Conserved His Residue of the Bacterial Sliding Clamp
Guillaume Compain, Clément Monsarrat, Julie Blagojevic, et al.
JACS Au (2024) Vol. 4, Iss. 2, pp. 432-440
Open Access | Times Cited: 8
Covalent hits and where to find them
Simon C. C. Lucas, J. Henry Blackwell, Sarah H. Hewitt, et al.
SLAS DISCOVERY (2024) Vol. 29, Iss. 3, pp. 100142-100142
Open Access | Times Cited: 7
Removing Neighboring Ring Influence in Monocyclic B–OH Diazaborines: Properties and Reactivity as Phenolic Bioisosteres with Dynamic Hydroxy Exchange
Jake J. Blackner, Olivia M. Schneider, Warren O. Wong, et al.
Journal of the American Chemical Society (2024) Vol. 146, Iss. 28, pp. 19499-19508
Closed Access | Times Cited: 6
Deciphering the enigmas of non‐nucleoside reverse transcriptase inhibitors (NNRTIs): A medicinal chemistry expedition towards combating HIV drug resistance
Kun Zhang, Yujie Zhang, Min Li, et al.
Medicinal Research Reviews (2024)
Closed Access | Times Cited: 6
Bioavailability, Biotransformation, and Excretion of the Covalent Bruton Tyrosine Kinase Inhibitor Acalabrutinib in Rats, Dogs, and Humans
Terry Podoll, Paul G. Pearson, Jerry Evarts, et al.
Drug Metabolism and Disposition (2018) Vol. 47, Iss. 2, pp. 145-154
Open Access | Times Cited: 58
How Reactive are Druggable Cysteines in Protein Kinases?
Ernest Awoonor‐Williams, Christopher N. Rowley
Journal of Chemical Information and Modeling (2018) Vol. 58, Iss. 9, pp. 1935-1946
Open Access | Times Cited: 54
Covalent Docking Identifies a Potent and Selective MKK7 Inhibitor
Amit Shraga, Evgenia Olshvang, Natalia Davidzohn, et al.
Cell chemical biology (2018) Vol. 26, Iss. 1, pp. 98-108.e5
Open Access | Times Cited: 54
Machine learning-accelerated quantum mechanics-based atomistic simulations for industrial applications
Tobias Morawietz, Nongnuch Artrith
Journal of Computer-Aided Molecular Design (2020) Vol. 35, Iss. 4, pp. 557-586
Open Access | Times Cited: 49
Aryl-fluorosulfate-based Lysine Covalent Pan-Inhibitors of Apoptosis Protein (IAP) Antagonists with Cellular Efficacy
Carlo Baggio, Parima Udompholkul, Luca Gambini, et al.
Journal of Medicinal Chemistry (2019) Vol. 62, Iss. 20, pp. 9188-9200
Open Access | Times Cited: 48
Mix-and-inject XFEL crystallography reveals gated conformational dynamics during enzyme catalysis.
Medhanjali Dasgupta, Dominik Budday, Saulo H. P. de Oliveira, et al.
Proceedings of the National Academy of Sciences (2019) Vol. 116, Iss. 51, pp. 25634-25640
Closed Access | Times Cited: 47
Itaconate is a covalent inhibitor of the Mycobacterium tuberculosis isocitrate lyase
Brooke X. C. Kwai, Annabelle J. Collins, Martin Middleditch, et al.
RSC Medicinal Chemistry (2020) Vol. 12, Iss. 1, pp. 57-61
Open Access | Times Cited: 46
How the Local Environment of Functional Sites Regulates Protein Function
Karine Mazmanian, Karen Sargsyan, Carmay Lim
Journal of the American Chemical Society (2020) Vol. 142, Iss. 22, pp. 9861-9871
Closed Access | Times Cited: 45
Toward the identification of ZDHHC enzymes required for palmitoylation of viral protein as potential drug targets
Mohamed Rasheed Gadalla, Michael Veit
Expert Opinion on Drug Discovery (2019) Vol. 15, Iss. 2, pp. 159-177
Closed Access | Times Cited: 44
Affinity and Selectivity Assessment of Covalent Inhibitors by Free Energy Calculations
Levente M. Mihalovits, György G. Ferenczy, György M. Keserű
Journal of Chemical Information and Modeling (2020) Vol. 60, Iss. 12, pp. 6579-6594
Closed Access | Times Cited: 40
Mechanism of covalent binding of ibrutinib to Bruton's tyrosine kinase revealed by QM/MM calculations
Angus Voice, Gary Tresadern, Rebecca M. Twidale, et al.
Chemical Science (2021) Vol. 12, Iss. 15, pp. 5511-5516
Open Access | Times Cited: 39

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