
OpenAlex is a bibliographic catalogue of scientific papers, authors and institutions accessible in open access mode, named after the Library of Alexandria. It's citation coverage is excellent and I hope you will find utility in this listing of citing articles!
If you click the article title, you'll navigate to the article, as listed in CrossRef. If you click the Open Access links, you'll navigate to the "best Open Access location". Clicking the citation count will open this listing for that article. Lastly at the bottom of the page, you'll find basic pagination options.
Requested Article:
Covalent drugs targeting histidine – an unexploited opportunity?
Jianwei Che, Lyn H. Jones
RSC Medicinal Chemistry (2022) Vol. 13, Iss. 10, pp. 1121-1126
Open Access | Times Cited: 31
Jianwei Che, Lyn H. Jones
RSC Medicinal Chemistry (2022) Vol. 13, Iss. 10, pp. 1121-1126
Open Access | Times Cited: 31
Showing 1-25 of 31 citing articles:
Emerging and Re-emerging Warheads for Targeted Covalent Inhibitors: An Update
Laura Hillebrand, Xiaojun Julia Liang, Ricardo A. M. Serafim, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 10, pp. 7668-7758
Closed Access | Times Cited: 49
Laura Hillebrand, Xiaojun Julia Liang, Ricardo A. M. Serafim, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 10, pp. 7668-7758
Closed Access | Times Cited: 49
Efficient Ligand Discovery Using Sulfur(VI) Fluoride Reactive Fragments
Arron Aatkar, Aini Vuorinen, Oliver Longfield, et al.
ACS Chemical Biology (2023) Vol. 18, Iss. 9, pp. 1926-1937
Open Access | Times Cited: 24
Arron Aatkar, Aini Vuorinen, Oliver Longfield, et al.
ACS Chemical Biology (2023) Vol. 18, Iss. 9, pp. 1926-1937
Open Access | Times Cited: 24
The expanding repertoire of covalent warheads for drug discovery
Namrashee V. Mehta, Mariam S. Degani
Drug Discovery Today (2023) Vol. 28, Iss. 12, pp. 103799-103799
Closed Access | Times Cited: 21
Namrashee V. Mehta, Mariam S. Degani
Drug Discovery Today (2023) Vol. 28, Iss. 12, pp. 103799-103799
Closed Access | Times Cited: 21
Development of a covalent cereblon-based PROTAC employing a fluorosulfate warhead
Radosław P. Nowak, Leah Ragosta, Fidel Huerta, et al.
RSC Chemical Biology (2023) Vol. 4, Iss. 11, pp. 906-912
Open Access | Times Cited: 20
Radosław P. Nowak, Leah Ragosta, Fidel Huerta, et al.
RSC Chemical Biology (2023) Vol. 4, Iss. 11, pp. 906-912
Open Access | Times Cited: 20
Peptide-Based Covalent Inhibitors Bearing Mild Electrophiles to Target a Conserved His Residue of the Bacterial Sliding Clamp
Guillaume Compain, Clément Monsarrat, Julie Blagojevic, et al.
JACS Au (2024) Vol. 4, Iss. 2, pp. 432-440
Open Access | Times Cited: 8
Guillaume Compain, Clément Monsarrat, Julie Blagojevic, et al.
JACS Au (2024) Vol. 4, Iss. 2, pp. 432-440
Open Access | Times Cited: 8
Covalent hits and where to find them
Simon C. C. Lucas, J. Henry Blackwell, Sarah H. Hewitt, et al.
SLAS DISCOVERY (2024) Vol. 29, Iss. 3, pp. 100142-100142
Open Access | Times Cited: 7
Simon C. C. Lucas, J. Henry Blackwell, Sarah H. Hewitt, et al.
SLAS DISCOVERY (2024) Vol. 29, Iss. 3, pp. 100142-100142
Open Access | Times Cited: 7
Covalent drug discovery using sulfur(VI) fluoride exchange warheads
Huang Huang, Lyn H. Jones
Expert Opinion on Drug Discovery (2023) Vol. 18, Iss. 7, pp. 725-735
Closed Access | Times Cited: 13
Huang Huang, Lyn H. Jones
Expert Opinion on Drug Discovery (2023) Vol. 18, Iss. 7, pp. 725-735
Closed Access | Times Cited: 13
Histidine-Covalent Stapled Alpha-Helical Peptides Targeting hMcl-1
Giulia Alboreggia, Parima Udompholkul, Carlo Baggio, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 10, pp. 8172-8185
Open Access | Times Cited: 4
Giulia Alboreggia, Parima Udompholkul, Carlo Baggio, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 10, pp. 8172-8185
Open Access | Times Cited: 4
Identification of an Allene Warhead That Selectively Targets a Histidine Residue in the Escherichia coli Oxidoreductase Enzyme DsbA
Yildiz Tasdan, Gautham R. Balaji, Naureen Akhtar, et al.
ACS Medicinal Chemistry Letters (2025)
Closed Access
Yildiz Tasdan, Gautham R. Balaji, Naureen Akhtar, et al.
ACS Medicinal Chemistry Letters (2025)
Closed Access
Covalent Stapling of the Cereblon Sensor Loop Histidine Using Sulfur-Heterocycle Exchange
Justin T. Cruite, Radosław P. Nowak, Katherine A. Donovan, et al.
ACS Medicinal Chemistry Letters (2023) Vol. 14, Iss. 11, pp. 1576-1581
Closed Access | Times Cited: 10
Justin T. Cruite, Radosław P. Nowak, Katherine A. Donovan, et al.
ACS Medicinal Chemistry Letters (2023) Vol. 14, Iss. 11, pp. 1576-1581
Closed Access | Times Cited: 10
Ligand discovery by activity-based protein profiling
Micah J. Niphakis, Benjamin F. Cravatt
Cell chemical biology (2024) Vol. 31, Iss. 9, pp. 1636-1651
Closed Access | Times Cited: 3
Micah J. Niphakis, Benjamin F. Cravatt
Cell chemical biology (2024) Vol. 31, Iss. 9, pp. 1636-1651
Closed Access | Times Cited: 3
Covalent Targeting of Histidine Residues with Aryl Fluorosulfates: Application to Mcl-1 BH3 Mimetics
Giulia Alboreggia, Parima Udompholkul, Emma L. Atienza, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 22, pp. 20214-20223
Open Access | Times Cited: 3
Giulia Alboreggia, Parima Udompholkul, Emma L. Atienza, et al.
Journal of Medicinal Chemistry (2024) Vol. 67, Iss. 22, pp. 20214-20223
Open Access | Times Cited: 3
Recent highlights in covalent inhibitor design
Kristen A. Marino, Robert Nicewonger, Hailong Zhang, et al.
Elsevier eBooks (2025)
Closed Access
Kristen A. Marino, Robert Nicewonger, Hailong Zhang, et al.
Elsevier eBooks (2025)
Closed Access
Covalent fragment approaches targeting non-cysteine residues
Noémi Csorba, Péter Ábrányi‐Balogh, György M. Keserű
Trends in Pharmacological Sciences (2023) Vol. 44, Iss. 11, pp. 802-816
Open Access | Times Cited: 7
Noémi Csorba, Péter Ábrányi‐Balogh, György M. Keserű
Trends in Pharmacological Sciences (2023) Vol. 44, Iss. 11, pp. 802-816
Open Access | Times Cited: 7
Activation-Free Sulfonyl Fluoride Probes for Fragment Screening
László Petri, Péter Ábrányi‐Balogh, Noémi Csorba, et al.
Molecules (2023) Vol. 28, Iss. 7, pp. 3042-3042
Open Access | Times Cited: 5
László Petri, Péter Ábrányi‐Balogh, Noémi Csorba, et al.
Molecules (2023) Vol. 28, Iss. 7, pp. 3042-3042
Open Access | Times Cited: 5
Novel partially reversible NDM-1 inhibitors based on the naturally occurring houttuynin
Lifang Wang, Yaowen Liang, Pan Luo, et al.
Bioorganic Chemistry (2024) Vol. 147, pp. 107328-107328
Closed Access | Times Cited: 1
Lifang Wang, Yaowen Liang, Pan Luo, et al.
Bioorganic Chemistry (2024) Vol. 147, pp. 107328-107328
Closed Access | Times Cited: 1
Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX
Aivaras Vaškevičius, Denis Baronas, Ja̅nis Leita̅ns, et al.
eLife (2024) Vol. 13
Open Access | Times Cited: 1
Aivaras Vaškevičius, Denis Baronas, Ja̅nis Leita̅ns, et al.
eLife (2024) Vol. 13
Open Access | Times Cited: 1
Advances in Activity‐Based Protein Profiling of Functional Tyrosines in Proteomes
Jeffrey W. Brulet, Anthony M. Ciancone, Kun Yuan, et al.
Israel Journal of Chemistry (2023) Vol. 63, Iss. 3-4
Open Access | Times Cited: 3
Jeffrey W. Brulet, Anthony M. Ciancone, Kun Yuan, et al.
Israel Journal of Chemistry (2023) Vol. 63, Iss. 3-4
Open Access | Times Cited: 3
Development of sulfonyl fluoride chemical probes to advance the discovery of cereblon modulators
Yingpeng Liu, Radosław P. Nowak, Jianwei Che, et al.
RSC Medicinal Chemistry (2024) Vol. 15, Iss. 2, pp. 607-611
Closed Access
Yingpeng Liu, Radosław P. Nowak, Jianwei Che, et al.
RSC Medicinal Chemistry (2024) Vol. 15, Iss. 2, pp. 607-611
Closed Access
His-Tagging: Exploring Precise Chemical Modification of Histidine-Containing Bioactive Peptide Sequences
Sourav Chatterjee, Bishwajit Paul, Govindaswamy Shanker
Synlett (2024)
Closed Access
Sourav Chatterjee, Bishwajit Paul, Govindaswamy Shanker
Synlett (2024)
Closed Access
Synthetic modification of protein surfaces to mediate induced-proximity pharmacology
Lyn H. Jones
RSC Medicinal Chemistry (2024) Vol. 15, Iss. 9, pp. 2974-2979
Closed Access
Lyn H. Jones
RSC Medicinal Chemistry (2024) Vol. 15, Iss. 9, pp. 2974-2979
Closed Access
Mass Spectrometry and Chemical Biology Approaches for Deconvoluting Epigenetic Targets
Antony J. Burton, Ghaith M. Hamza, Anthony A. Iannetta, et al.
Royal Society of Chemistry eBooks (2024), pp. 50-83
Closed Access
Antony J. Burton, Ghaith M. Hamza, Anthony A. Iannetta, et al.
Royal Society of Chemistry eBooks (2024), pp. 50-83
Closed Access
Covalent Inhibitors of MAP Kinases
Surya K. De
Drug design and discovery (2024), pp. 159-189
Closed Access
Surya K. De
Drug design and discovery (2024), pp. 159-189
Closed Access
Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX
Aivaras Vaškevičius, Denis Baronas, Ja̅nis Leita̅ns, et al.
bioRxiv (Cold Spring Harbor Laboratory) (2024)
Open Access
Aivaras Vaškevičius, Denis Baronas, Ja̅nis Leita̅ns, et al.
bioRxiv (Cold Spring Harbor Laboratory) (2024)
Open Access
Covalent Inhibition of a Host–Pathogen Protein–Protein Interaction Reduces the Infectivity of Streptococcus pneumoniae
Yuhan Lyu, Fan Yang, Bharathi Sundaresh, et al.
JACS Au (2024) Vol. 4, Iss. 7, pp. 2484-2491
Open Access
Yuhan Lyu, Fan Yang, Bharathi Sundaresh, et al.
JACS Au (2024) Vol. 4, Iss. 7, pp. 2484-2491
Open Access